Once you have completed your screening procedure, what is the next step? This eBook outlines how biochemical assays are used to characterize and prioritize compounds following a primary screen of an enzyme target, whether through high throughput screening (HTS) or virtual screening (VS).
This eBook will outline key strategies for hit-to-lead selection, including:
- Assay Considerations
- Compound Triaging
- Hit Confirmation
- Hit Expansion
- Mechanism of Action Studies
- Residence Time Measurement
- Running a Dose-Response
Download the full eBook now to learn more
About BellBrook Labs
BellBrook Labs is dedicated to providing the pharmaceutical industry with enabling screening tools to accelerate the discovery of more effective therapies. Leveraging its two base platforms, BellBrook has developed assays for hundreds of drug targets.